Structure–ativity relationship of adenosine 5′-diphosphoribose at the transient receptor potential melastatin 2 (TRPM2) channel: rational design of antagonists

Christelle Moreau; Tanja Kirchberger; Joanna M. Swarbrick; Stephen J. Bartlett; Ralf Fliegert; Timur Yorgan; Andreas Bauche; Angelika Harneit; Andreas H. Guse; Barry V. L. Potter

doi:10.1021/jm401497a

Structure–ativity relationship of adenosine 5′-diphosphoribose at the transient receptor potential melastatin 2 (TRPM2) channel: rational design of antagonists

Christelle Moreau
, Tanja Kirchberger
, Joanna M. Swarbrick
, Stephen J. Bartlett
, Ralf Fliegert
, Timur Yorgan
, Andreas Bauche
, Angelika Harneit
, Andreas H. Guse
, Barry V. L. Potter

Department of Life Sciences

University Medical Centre Hamburg-Eppendorf

Research output: Contribution to journal › Article › peer-review

66 Citations (SciVal)

Original language	English
Pages (from-to)	10079-10102
Journal	Journal of Medicinal Chemistry
Volume	56
Issue number	24
DOIs	https://doi.org/10.1021/jm401497a
Publication status	Published - 27 Dec 2013

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10.1021/jm401497a

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Moreau, C., Kirchberger, T., Swarbrick, J. M., Bartlett, S. J., Fliegert, R., Yorgan, T., Bauche, A., Harneit, A., Guse, A. H., & Potter, B. V. L. (2013). Structure–ativity relationship of adenosine 5′-diphosphoribose at the transient receptor potential melastatin 2 (TRPM2) channel: rational design of antagonists. Journal of Medicinal Chemistry, 56(24), 10079-10102. https://doi.org/10.1021/jm401497a

Structure–ativity relationship of adenosine 5′-diphosphoribose at the transient receptor potential melastatin 2 (TRPM2) channel: rational design of antagonists. / Moreau, Christelle; Kirchberger, Tanja; Swarbrick, Joanna M. et al.
In: Journal of Medicinal Chemistry, Vol. 56, No. 24, 27.12.2013, p. 10079-10102.

Research output: Contribution to journal › Article › peer-review

Moreau, C, Kirchberger, T, Swarbrick, JM, Bartlett, SJ, Fliegert, R, Yorgan, T, Bauche, A, Harneit, A, Guse, AH & Potter, BVL 2013, 'Structure–ativity relationship of adenosine 5′-diphosphoribose at the transient receptor potential melastatin 2 (TRPM2) channel: rational design of antagonists', Journal of Medicinal Chemistry, vol. 56, no. 24, pp. 10079-10102. https://doi.org/10.1021/jm401497a

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author = "Christelle Moreau and Tanja Kirchberger and Swarbrick, \{Joanna M.\} and Bartlett, \{Stephen J.\} and Ralf Fliegert and Timur Yorgan and Andreas Bauche and Angelika Harneit and Guse, \{Andreas H.\} and Potter, \{Barry V. L.\}",

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Structure–ativity relationship of adenosine 5′-diphosphoribose at the transient receptor potential melastatin 2 (TRPM2) channel: rational design of antagonists

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