Selective formation of 1,3-oxazolidine-2-thiones on ketohexose templates

A Tatibouet, S Lawrence, P Rollin, G D Holman

Research output: Contribution to journalArticle

17 Citations (Scopus)

Abstract

Thiocyanic acid condensation on selectively protected ketohexose led to the isolation of five out of the seven possible 1,3-oxazolidine-2-thiones (OZT). The four isomeric spiro-OZT synthesized showed promising biological activity against D-fructose transport.
Original languageEnglish
Pages (from-to)1945-1948
Number of pages4
JournalSynlett
Issue number11
DOIs
Publication statusPublished - 2004

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Thiones
Bioactivity
Fructose
Condensation
oxazolidine
spiro-oxazolidine
thiocyanic acid

Cite this

Selective formation of 1,3-oxazolidine-2-thiones on ketohexose templates. / Tatibouet, A; Lawrence, S; Rollin, P; Holman, G D.

In: Synlett, No. 11, 2004, p. 1945-1948.

Research output: Contribution to journalArticle

Tatibouet, A ; Lawrence, S ; Rollin, P ; Holman, G D. / Selective formation of 1,3-oxazolidine-2-thiones on ketohexose templates. In: Synlett. 2004 ; No. 11. pp. 1945-1948.
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