Opioid binding and  in vitro  profiles of a series of 4-hydroxy-3-methoxyindolomorphinans. Transformation of a δ-selective ligand into a high affinity  k -selective ligand by introduction of a 5,14-substituted bridge

P Grundt; F Martinez-Bermejo; J W Lewis; S M Husbands

Opioid binding and in vitro profiles of a series of 4-hydroxy-3-methoxyindolomorphinans. Transformation of a δ-selective ligand into a high affinity k -selective ligand by introduction of a 5,14-substituted bridge

P Grundt
, F Martinez-Bermejo
, J W Lewis
, S M Husbands

Department of Life Sciences

Research output: Contribution to journal › Article › peer-review

10 Citations (SciVal)

Original language	English
Pages (from-to)	3174-3177
Number of pages	4
Journal	Journal of Medicinal Chemistry
Volume	46
Publication status	Published - 2003

Keywords

in vitro

Cite this

Opioid binding and in vitro profiles of a series of 4-hydroxy-3-methoxyindolomorphinans. Transformation of a δ-selective ligand into a high affinity k -selective ligand by introduction of a 5,14-substituted bridge. / Grundt, P; Martinez-Bermejo, F; Lewis, J W et al.
In: Journal of Medicinal Chemistry, Vol. 46, 2003, p. 3174-3177.

Research output: Contribution to journal › Article › peer-review

@article{68ade8465e9f4a36b17f468ad1fb26ef,

title = "Opioid binding and in vitro profiles of a series of 4-hydroxy-3-methoxyindolomorphinans. Transformation of a δ-selective ligand into a high affinity k -selective ligand by introduction of a 5,14-substituted bridge",

keywords = "in vitro",

author = "P Grundt and F Martinez-Bermejo and Lewis, \{J W\} and Husbands, \{S M\}",

year = "2003",

language = "English",

volume = "46",

pages = "3174--3177",

journal = "Journal of Medicinal Chemistry",

issn = "0022-2623",

publisher = "American Chemical Society",

}

TY - JOUR

T1 - Opioid binding and in vitro profiles of a series of 4-hydroxy-3-methoxyindolomorphinans. Transformation of a δ-selective ligand into a high affinity k -selective ligand by introduction of a 5,14-substituted bridge

AU - Grundt, P

AU - Martinez-Bermejo, F

AU - Lewis, J W

AU - Husbands, S M

PY - 2003

Y1 - 2003

KW - in vitro

M3 - Article

SN - 0022-2623

VL - 46

SP - 3174

EP - 3177

JO - Journal of Medicinal Chemistry

JF - Journal of Medicinal Chemistry

ER -