Opioid binding and  in vitro  profiles of a series of 4-hydroxy-3-methoxyindolomorphinans. Transformation of a δ-selective ligand into a high affinity  k -selective ligand by introduction of a 5,14-substituted bridge

P Grundt; F Martinez-Bermejo; J W Lewis; S M Husbands

Opioid binding and in vitro profiles of a series of 4-hydroxy-3-methoxyindolomorphinans. Transformation of a δ-selective ligand into a high affinity k -selective ligand by introduction of a 5,14-substituted bridge

P Grundt, F Martinez-Bermejo, J W Lewis, S M Husbands

Department of Life Sciences

Research output: Contribution to journal › Article › peer-review

10 Citations (SciVal)

Original language	English
Pages (from-to)	3174-3177
Number of pages	4
Journal	Journal of Medicinal Chemistry
Volume	46
Publication status	Published - 2003

Keywords

in vitro

Cite this

Opioid binding and in vitro profiles of a series of 4-hydroxy-3-methoxyindolomorphinans. Transformation of a δ-selective ligand into a high affinity k -selective ligand by introduction of a 5,14-substituted bridge. / Grundt, P; Martinez-Bermejo, F; Lewis, J W et al.
In: Journal of Medicinal Chemistry, Vol. 46, 2003, p. 3174-3177.

Research output: Contribution to journal › Article › peer-review

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AU - Grundt, P

AU - Martinez-Bermejo, F

AU - Lewis, J W

AU - Husbands, S M

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