Novel Aryl and Heteroaryl Acyl Sulfamide Synthesis via Microwave-Assisted Palladium-Catalyzed Carbonylation

Bryan Roberts; David Liptrot; Lilian Alcaraz

doi:10.1021/ol100083w

Novel Aryl and Heteroaryl Acyl Sulfamide Synthesis via Microwave-Assisted Palladium-Catalyzed Carbonylation

Bryan Roberts, David Liptrot, Lilian Alcaraz

Department of Chemistry

Research output: Contribution to journal › Article › peer-review

17 Citations (SciVal)

Abstract

A novel, simple synthesis of aryl and heteroaryl acyl sulfamides has been developed via palladium-catalyzed carbonylation of aryl or heteroaryl halides in the presence of sulfamide nucleophiles. A range of reactions illustrating the wide scope of this reaction was carried out under microwave irradiation in a vessel equipped with a gas inlet adapter and proceeded in good to excellent yields.

Original language	English
Pages (from-to)	1264-1267
Number of pages	4
Journal	Organic Letters
Volume	12
Issue number	6
DOIs	https://doi.org/10.1021/ol100083w
Publication status	Published - 19 Mar 2010

Access to Document

10.1021/ol100083w

Cite this

@article{bc069b83f7d048db92a4bfd8b5158f27,

title = "Novel Aryl and Heteroaryl Acyl Sulfamide Synthesis via Microwave-Assisted Palladium-Catalyzed Carbonylation",

abstract = "A novel, simple synthesis of aryl and heteroaryl acyl sulfamides has been developed via palladium-catalyzed carbonylation of aryl or heteroaryl halides in the presence of sulfamide nucleophiles. A range of reactions illustrating the wide scope of this reaction was carried out under microwave irradiation in a vessel equipped with a gas inlet adapter and proceeded in good to excellent yields.",

author = "Bryan Roberts and David Liptrot and Lilian Alcaraz",

year = "2010",

month = mar,

day = "19",

doi = "10.1021/ol100083w",

language = "English",

volume = "12",

pages = "1264--1267",

journal = "Organic Letters",

issn = "1523-7060",

publisher = "American Chemical Society",

number = "6",

}

TY - JOUR

T1 - Novel Aryl and Heteroaryl Acyl Sulfamide Synthesis via Microwave-Assisted Palladium-Catalyzed Carbonylation

AU - Roberts, Bryan

AU - Liptrot, David

AU - Alcaraz, Lilian

PY - 2010/3/19

Y1 - 2010/3/19

N2 - A novel, simple synthesis of aryl and heteroaryl acyl sulfamides has been developed via palladium-catalyzed carbonylation of aryl or heteroaryl halides in the presence of sulfamide nucleophiles. A range of reactions illustrating the wide scope of this reaction was carried out under microwave irradiation in a vessel equipped with a gas inlet adapter and proceeded in good to excellent yields.

AB - A novel, simple synthesis of aryl and heteroaryl acyl sulfamides has been developed via palladium-catalyzed carbonylation of aryl or heteroaryl halides in the presence of sulfamide nucleophiles. A range of reactions illustrating the wide scope of this reaction was carried out under microwave irradiation in a vessel equipped with a gas inlet adapter and proceeded in good to excellent yields.

U2 - 10.1021/ol100083w

DO - 10.1021/ol100083w

M3 - Article

VL - 12

SP - 1264

EP - 1267

JO - Organic Letters

JF - Organic Letters

SN - 1523-7060

IS - 6

ER -

Novel Aryl and Heteroaryl Acyl Sulfamide Synthesis via Microwave-Assisted Palladium-Catalyzed Carbonylation

Abstract

Access to Document

Fingerprint

Cite this