Iterative amination strategy in the synthesis of peptidomimetics

C.G. Frost, P. Mendonça

Research output: Contribution to journalArticle

7 Citations (Scopus)

Abstract

An iterative palladium catalysed cross-coupling reaction of aryl bromides with amines has been employed in the preparation of novel peptidomimetics. This is a versatile strategy with which we can demonstrate the principle of library synthesis by using a diverse range of coupling partners.
Original languageEnglish
Pages (from-to)1159-1160
Number of pages2
JournalChemistry Letters
Volume26
Issue number11
DOIs
Publication statusPublished - 1997

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Peptidomimetics
Amination
Palladium
Bromides
Amines

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Iterative amination strategy in the synthesis of peptidomimetics. / Frost, C.G.; Mendonça, P.

In: Chemistry Letters, Vol. 26, No. 11, 1997, p. 1159-1160.

Research output: Contribution to journalArticle

Frost, C.G. ; Mendonça, P. / Iterative amination strategy in the synthesis of peptidomimetics. In: Chemistry Letters. 1997 ; Vol. 26, No. 11. pp. 1159-1160.
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