Formyloxyacetoxyphenylmethane as an N-Formylating Reagent for Amines, Amino Acids, and Peptides

Robert Chapman; Ruth Lawrence; Jonathan Williams; Steven Bull

doi:10.1021/acs.orglett.7b02382

Formyloxyacetoxyphenylmethane as an N-Formylating Reagent for Amines, Amino Acids, and Peptides

Robert Chapman, Ruth Lawrence, Jonathan Williams, Steven Bull

Research output: Contribution to conference › Paper › peer-review

27 Citations (SciVal)

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Abstract

Formyloxyacetoxyphenylmethane is a stable, water-tolerant, N-formylating reagent for primary and secondary amines that can be used under solvent-free conditions at room temperature to prepare a range of N-formamides, N-formylanilines, N-formyl-α-amino acids, N-formylpeptides, and an isocyanide.

Original language	English
Pages	4908-4911
DOIs	https://doi.org/10.1021/acs.orglett.7b02382
Publication status	Published - 30 Aug 2017

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10.1021/acs.orglett.7b02382

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title = "Formyloxyacetoxyphenylmethane as an N-Formylating Reagent for Amines, Amino Acids, and Peptides",

abstract = "Formyloxyacetoxyphenylmethane is a stable, water-tolerant, N-formylating reagent for primary and secondary amines that can be used under solvent-free conditions at room temperature to prepare a range of N-formamides, N-formylanilines, N-formyl-α-amino acids, N-formylpeptides, and an isocyanide.",

author = "Robert Chapman and Ruth Lawrence and Jonathan Williams and Steven Bull",

year = "2017",

month = aug,

day = "30",

doi = "10.1021/acs.orglett.7b02382",

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T1 - Formyloxyacetoxyphenylmethane as an N-Formylating Reagent for Amines, Amino Acids, and Peptides

AU - Chapman, Robert

AU - Lawrence, Ruth

AU - Williams, Jonathan

AU - Bull, Steven

PY - 2017/8/30

Y1 - 2017/8/30

N2 - Formyloxyacetoxyphenylmethane is a stable, water-tolerant, N-formylating reagent for primary and secondary amines that can be used under solvent-free conditions at room temperature to prepare a range of N-formamides, N-formylanilines, N-formyl-α-amino acids, N-formylpeptides, and an isocyanide.

AB - Formyloxyacetoxyphenylmethane is a stable, water-tolerant, N-formylating reagent for primary and secondary amines that can be used under solvent-free conditions at room temperature to prepare a range of N-formamides, N-formylanilines, N-formyl-α-amino acids, N-formylpeptides, and an isocyanide.

UR - http://pubs.acs.org/doi/10.1021/acs.orglett.7b02382

U2 - 10.1021/acs.orglett.7b02382

DO - 10.1021/acs.orglett.7b02382

M3 - Paper

SP - 4908

EP - 4911

ER -

Formyloxyacetoxyphenylmethane as an N-Formylating Reagent for Amines, Amino Acids, and Peptides

Abstract

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