Dual aromatase-sulfatase inhibitors based on the anastrozole template: synthesis, in vitro SAR, molecular modelling and in vivo activity

Toby Jackson; L. W. Lawrence Woo; Melanie N. Trusselle; Surinder K. Chander; Atul Purohit; Michael J. Reed; Barry V. L. Potter

doi:10.1039/B707768H

Dual aromatase-sulfatase inhibitors based on the anastrozole template: synthesis, in vitro SAR, molecular modelling and in vivo activity

Toby Jackson
, L. W. Lawrence Woo
, Melanie N. Trusselle
, Surinder K. Chander
, Atul Purohit
, Michael J. Reed
, Barry V. L. Potter

Department of Life Sciences

Research output: Contribution to journal › Article › peer-review

66 Citations (SciVal)

Original language	English
Pages (from-to)	2940-2952
Journal	Organic and Biomolecular Chemistry
Volume	5
DOIs	https://doi.org/10.1039/B707768H
Publication status	Published - 2007

Keywords

in vitro

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10.1039/B707768H

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title = "Dual aromatase-sulfatase inhibitors based on the anastrozole template: synthesis, in vitro SAR, molecular modelling and in vivo activity",

keywords = "in vitro",

author = "Toby Jackson and Woo, \{L. W. Lawrence\} and Trusselle, \{Melanie N.\} and Chander, \{Surinder K.\} and Atul Purohit and Reed, \{Michael J.\} and Potter, \{Barry V. L.\}",

year = "2007",

doi = "10.1039/B707768H",

language = "English",

volume = "5",

pages = "2940--2952",

journal = "Organic and Biomolecular Chemistry",

issn = "1477-0520",

publisher = "Royal Society of Chemistry",

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TY - JOUR

T1 - Dual aromatase-sulfatase inhibitors based on the anastrozole template

T2 - synthesis, in vitro SAR, molecular modelling and in vivo activity

AU - Jackson, Toby

AU - Woo, L. W. Lawrence

AU - Trusselle, Melanie N.

AU - Chander, Surinder K.

AU - Purohit, Atul

AU - Reed, Michael J.

AU - Potter, Barry V. L.

PY - 2007

Y1 - 2007

KW - in vitro

UR - http://dx.doi.org/10.1039/B707768H

U2 - 10.1039/B707768H

DO - 10.1039/B707768H

M3 - Article

SN - 1477-0520

VL - 5

SP - 2940

EP - 2952

JO - Organic and Biomolecular Chemistry

JF - Organic and Biomolecular Chemistry

ER -

Dual aromatase-sulfatase inhibitors based on the anastrozole template: synthesis, in vitro SAR, molecular modelling and in vivo activity

Keywords

Access to Document

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