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BU08073 a buprenorphine analog with partial agonist activity at μ-receptors in vitro but long-lasting opioid antagonist activity in vivo in mice

T. V. Khroyan, J. Wu, W. E. Polgar, G. Cami-Kobeci, N. Fotaki, Stephen M. Husbands, Lawrence Toll

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Pharmacology, Toxicology and Pharmaceutical Science