Anticancer steroid sulfatase inhibitors

synthesis of a potent fluorinated second-generation agent, in vitro and in vivo activities, molecular modeling, and protein crystallography

L. W. Lawrence Woo, Delphine S. Fischer, Christopher M. Sharland, Melanie Trusselle, Paul A. Foster, Surinder K. Chander, Anna Di Fiore, Claudiu T. Supuran, Giuseppina De Simone, Atul Purohit, Michael J. Reed, Barry V. L. Potter

Research output: Contribution to journalArticle

33 Citations (Scopus)
Original languageEnglish
Pages (from-to)2435-2444
JournalMolecular Cancer Therapeutics
Volume7
Issue number8
DOIs
Publication statusPublished - 2008

Cite this

Anticancer steroid sulfatase inhibitors : synthesis of a potent fluorinated second-generation agent, in vitro and in vivo activities, molecular modeling, and protein crystallography. / Woo, L. W. Lawrence; Fischer, Delphine S.; Sharland, Christopher M.; Trusselle, Melanie; Foster, Paul A.; Chander, Surinder K.; Di Fiore, Anna; Supuran, Claudiu T.; De Simone, Giuseppina; Purohit, Atul; Reed, Michael J.; Potter, Barry V. L.

In: Molecular Cancer Therapeutics, Vol. 7, No. 8, 2008, p. 2435-2444.

Research output: Contribution to journalArticle

Woo, LWL, Fischer, DS, Sharland, CM, Trusselle, M, Foster, PA, Chander, SK, Di Fiore, A, Supuran, CT, De Simone, G, Purohit, A, Reed, MJ & Potter, BVL 2008, 'Anticancer steroid sulfatase inhibitors: synthesis of a potent fluorinated second-generation agent, in vitro and in vivo activities, molecular modeling, and protein crystallography', Molecular Cancer Therapeutics, vol. 7, no. 8, pp. 2435-2444. https://doi.org/10.1158/1535-7163.MCT-08-0195
Woo, L. W. Lawrence ; Fischer, Delphine S. ; Sharland, Christopher M. ; Trusselle, Melanie ; Foster, Paul A. ; Chander, Surinder K. ; Di Fiore, Anna ; Supuran, Claudiu T. ; De Simone, Giuseppina ; Purohit, Atul ; Reed, Michael J. ; Potter, Barry V. L. / Anticancer steroid sulfatase inhibitors : synthesis of a potent fluorinated second-generation agent, in vitro and in vivo activities, molecular modeling, and protein crystallography. In: Molecular Cancer Therapeutics. 2008 ; Vol. 7, No. 8. pp. 2435-2444.
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