1,1-Diacyloxy-1-phenylmethanes as versatile N-acylating agents for amines

Robert S.L. Chapman; Joshua D. Tibbetts; Steven D. Bull

doi:10.1016/j.tet.2018.05.044

1,1-Diacyloxy-1-phenylmethanes as versatile N-acylating agents for amines

Robert S.L. Chapman, Joshua D. Tibbetts, Steven D. Bull

Research output: Contribution to journal › Article › peer-review

3 Citations (SciVal)

45 Downloads (Pure)

Abstract

1,1-Diacyloxy-1-phenylmethanes and 1-pivaloxy-1-acyloxy-1-phenylmethanes have been used as bench stable N-acylating reagents for primary and secondary amines and anilines under solvent-free conditions to afford their corresponding amides in good yield.

Original language	English
Pages (from-to)	5330-5339
Number of pages	10
Journal	Tetrahedron
Volume	74
Issue number	38
Early online date	21 May 2018
DOIs	https://doi.org/10.1016/j.tet.2018.05.044
Publication status	Published - 20 Sep 2018

Keywords

1,1-Acylals
Amides
N-Acylation
Solvent free

ASJC Scopus subject areas

Biochemistry
Drug Discovery
Organic Chemistry

Access to Document

10.1016/j.tet.2018.05.044

1,1-Diacyloxy-1-Phenylmethanes as Versatile N-Acylating Agents for AminesAccepted author manuscript, 1.01 MBLicence: CC BY-NC-ND

Cite this

@article{73bd2f9efd8b4ab49b1ee75215550cdc,

title = "1,1-Diacyloxy-1-phenylmethanes as versatile N-acylating agents for amines",

abstract = "1,1-Diacyloxy-1-phenylmethanes and 1-pivaloxy-1-acyloxy-1-phenylmethanes have been used as bench stable N-acylating reagents for primary and secondary amines and anilines under solvent-free conditions to afford their corresponding amides in good yield.",

keywords = "1,1-Acylals, Amides, N-Acylation, Solvent free",

author = "Chapman, {Robert S.L.} and Tibbetts, {Joshua D.} and Bull, {Steven D.}",

year = "2018",

month = sep,

day = "20",

doi = "10.1016/j.tet.2018.05.044",

language = "English",

volume = "74",

pages = "5330--5339",

journal = "Tetrahedron",

issn = "0040-4020",

publisher = "Elsevier",

number = "38",

}

TY - JOUR

T1 - 1,1-Diacyloxy-1-phenylmethanes as versatile N-acylating agents for amines

AU - Chapman, Robert S.L.

AU - Tibbetts, Joshua D.

AU - Bull, Steven D.

PY - 2018/9/20

Y1 - 2018/9/20

N2 - 1,1-Diacyloxy-1-phenylmethanes and 1-pivaloxy-1-acyloxy-1-phenylmethanes have been used as bench stable N-acylating reagents for primary and secondary amines and anilines under solvent-free conditions to afford their corresponding amides in good yield.

AB - 1,1-Diacyloxy-1-phenylmethanes and 1-pivaloxy-1-acyloxy-1-phenylmethanes have been used as bench stable N-acylating reagents for primary and secondary amines and anilines under solvent-free conditions to afford their corresponding amides in good yield.

KW - 1,1-Acylals

KW - Amides

KW - N-Acylation

KW - Solvent free

UR - http://www.scopus.com/inward/record.url?scp=85048338873&partnerID=8YFLogxK

U2 - 10.1016/j.tet.2018.05.044

DO - 10.1016/j.tet.2018.05.044

M3 - Article

AN - SCOPUS:85048338873

VL - 74

SP - 5330

EP - 5339

JO - Tetrahedron

JF - Tetrahedron

SN - 0040-4020

IS - 38

ER -

1,1-Diacyloxy-1-phenylmethanes as versatile N-acylating agents for amines

Abstract

Keywords

ASJC Scopus subject areas

Access to Document

Other files and links

Fingerprint

Cite this