1,1-Diacyloxy-1-phenylmethanes as versatile N-acylating agents for amines

Robert S.L. Chapman; Joshua D. Tibbetts; Steven D. Bull

doi:10.1016/j.tet.2018.05.044

1,1-Diacyloxy-1-phenylmethanes as versatile N-acylating agents for amines

Robert S.L. Chapman, Joshua D. Tibbetts, Steven D. Bull

Research output: Contribution to journal › Article

2 Citations (Scopus)

28 Downloads (Pure)

Abstract

1,1-Diacyloxy-1-phenylmethanes and 1-pivaloxy-1-acyloxy-1-phenylmethanes have been used as bench stable N-acylating reagents for primary and secondary amines and anilines under solvent-free conditions to afford their corresponding amides in good yield.

Original language	English
Pages (from-to)	5330-5339
Number of pages	10
Journal	Tetrahedron
Volume	74
Issue number	38
Early online date	21 May 2018
DOIs	https://doi.org/10.1016/j.tet.2018.05.044
Publication status	Published - 20 Sep 2018

Keywords

1,1-Acylals
Amides
N-Acylation
Solvent free

ASJC Scopus subject areas

Biochemistry
Drug Discovery
Organic Chemistry

Access to Document

10.1016/j.tet.2018.05.044

1,1-Diacyloxy-1-Phenylmethanes as Versatile N-Acylating Agents for AminesAccepted author manuscript, 1.01 MBLicence: CC BY-NC-ND

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Chapman, R. S. L., Tibbetts, J. D., & Bull, S. D. (2018). 1,1-Diacyloxy-1-phenylmethanes as versatile N-acylating agents for amines. Tetrahedron, 74(38), 5330-5339. https://doi.org/10.1016/j.tet.2018.05.044

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