Research output
- 5 Article
Search results
-
2026
Molecular basis of domain-specific angiotensin I-converting enzyme inhibition by the antihypertensive drugs enalaprilat, ramiprilat, trandolaprilat, quinaprilat and perindoprilat
Gregory, K. S., Ramasamy, V., Sturrock, E. D. & Acharya, K. R., 31 Jan 2026, In: FEBS Journal. 293, 2, p. 475-491Research output: Contribution to journal › Article › peer-review
Open Access -
2025
Ciprofloxacin inhibits angiotensin I -converting enzyme (ACE) activity by binding at the exosite, distal to the catalytic pocket
Gregory, K. S., Ramasamy, V., Sturrock, E. D. & Acharya, K. R., 15 Oct 2025, In: ACS Bio & Med Chem Au. 5, 5, p. 852-859Research output: Contribution to journal › Article › peer-review
Open Access -
Design of Novel Mercapto-3-phenylpropanoyl Dipeptides as Dual Angiotensin-Converting Enzyme C-Domain-Selective/Neprilysin Inhibitors
Acharya, R., Sturrock, E., Cozier, G., Eyermann, C., Basarab, G., Schwager, S. L. U., Chibale, K. & Coulson, L., 10 Apr 2025, In: Journal of Medicinal Chemistry. 68, 7, p. 7720-7736 17 p.Research output: Contribution to journal › Article › peer-review
Open Access1 Link opens in a new tab Citation (SciVal) -
Molecular basis of human angiotensin-1 converting enzyme inhibition by a series of diprolyl-derived compounds
Gregory, K. S., Cozier, G. E., Fienberg, S., Chibale, K., Sturrock, E. D. & Acharya, R., 6 Jan 2025, (E-pub ahead of print) In: FEBS Journal.Research output: Contribution to journal › Article › peer-review
Open Access -
2024
Structural insights into the inhibitory mechanism of angiotensin-I converting enzyme by the lactotripeptides IPP and VPP
Gregory, K. S., Cozier, G. E., Schwager, S. L. U., Sturrock, E. D. & Acharya, K. R., 31 Jan 2024, In: FEBS Letters. 598, 2, p. 242-251 10 p.Research output: Contribution to journal › Article › peer-review
Open Access17 Link opens in a new tab Citations (SciVal)