Research output per year
Research output per year
- 10 results
Search results
-
2021
Racemases and epimerases operating through a 1,1-proton transfer mechanism: Reactivity, mechanism and inhibition
Lloyd, M., Jevglevskis, M., Nathubhai, A., James, T., Threadgill, M. & Woodman, T., 1 May 2021, In: Chemical Society Reviews. 50, 10, p. 5952–5984 33 p.Research output: Contribution to journal › Review article › peer-review
Open Access14 Citations (SciVal) -
2019
Identification of novel small-molecule inhibitors of α-methylacyl-CoA racemase (AMACR; P504S) and structure-activity relationships
Petrova, Y., Wadda, K., Nathubhai, A., Jevglevskis, M., Mitchell, P., James, T., Threadgill, M., Woodman, T. & Lloyd, M., 1 Nov 2019, In: Bioorganic Chemistry. 92, 103264.Research output: Contribution to journal › Article › peer-review
Open AccessFile12 Citations (SciVal)139 Downloads (Pure) -
Novel 2-arylthiopropanoyl-CoA inhibitors of α-methylacyl-CoA racemase 1A (AMACR; P504S) as potential anti-prostate cancer agents
Jevglevskis, M., Nathubhai, A., Wadda, K., Lee, G. L., Al-Rawi, S., Jiao, T., Mitchell, P., James, T., Threadgill, M., Woodman, T. & Lloyd, M., 1 Nov 2019, In: Bioorganic Chemistry. 92, 103263.Research output: Contribution to journal › Article › peer-review
Open AccessFile11 Citations (SciVal)252 Downloads (Pure) -
2018
Structure-activity relationships of rationally designed AMACR 1A inhibitors
Jevglevskis, M., Lee, G. L., Nathubhai, A., Petrova, Y., James, T., Threadgill, M., Woodman, T. & Lloyd, M., 1 Sept 2018, In: Bioorganic and Medicinal Chemistry. 79, p. 145-154 10 p.Research output: Contribution to journal › Article › peer-review
Open AccessFile9 Citations (SciVal)114 Downloads (Pure) -
2017
A convenient colorimetric assay for α-methylacyl-CoA racemase (AMACR; P504S) and testing of inhibitors
Jevglevskis, M., Lee, G. L., Nathubhai, A., James, T., Threadgill, M., Woodman, T. & Lloyd, M., 21 Apr 2017, (Unpublished).Research output: Contribution to conference › Abstract › peer-review
File73 Downloads (Pure) -
A novel colorimetric assay for α-methylacyl-CoA racemase 1A (AMACR; P504S) utilizing the elimination of 2,4-dinitrophenolate
Jevglevskis, M., Lee, G. L., Nathubhai, A., Petrova, Y., James, T., Threadgill, M., Woodman, T. & Lloyd, M., 7 May 2017, In: Chemical Communications. 53, 37, p. 5087-5090 4 p.Research output: Contribution to journal › Article › peer-review
Open Access18 Citations (SciVal) -
2016
A Convenient Colorimetric Assay For Alpha-Methylacyl-CoA Racemase (AMACR; P504S) And Testing Of Inhibitors
Jevglevskis, M., Lee, G. L., Nathubhai, A., Petrova, Y., Threadgill, M., James, T., Woodman, T. & Lloyd, M., Jun 2016.Research output: Contribution to conference › Poster
Open AccessFile65 Downloads (Pure) -
A Study On The α-Methylacyl-CoA Racemase (AMACR) Elimination Reaction And Its Application To Inhibitor Testing
Jevglevskis, M., Lee, G. L., Sun, J., Zhou, S., Sun, X., Kociok-Kohn, G., James, T., Woodman, T. & Lloyd, M., 27 Apr 2016, (Unpublished).Research output: Contribution to conference › Poster
File78 Downloads (Pure) -
2015
A Convenient Colorimetric Assay for α-Methylacyl-CoA Racemase (AMACR; P504S) and Testing Of Inhibitors
Jevglevskis, M., Lee, G. L., Nathubhai, A., James, T., Threadgill, M., Woodman, T. & Lloyd, M., 11 Nov 2015, (Unpublished).Research output: Contribution to conference › Poster
File67 Downloads (Pure) -
New routes to fight castrate-resistant prostate cancer: targeting α-methylacyl-CoA racemase (AMACR)
Lee, G. L., Jevglevskis, M., Threadgill, M., Woodman, T. & Lloyd, M., 2015.Research output: Contribution to conference › Poster › peer-review